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 Recent Publications (2002 - present)

  1. Bates RW, Sa-Ei K. O-alkenyl hydroxylamines: a new concept for cyclofunctionalization. Org Lett 2002;4:4225-7.
  2. Bates RW, Satcharoen V. Nucleophilic transition metal based cyclization of allenes. Chem Soc Rev 2002;31:12-21.
  3. Bates RW, Sa-Ei K. Syntheses of the sedum and related alkaloids. Tetrahedron 2002;58:5957-78.
  4. Chuankamnerdkarn M, Sutthivaiyakit S, Thasana N, Pisutjaroenpong S. Prenylated isoflavones from Derris scandens. Heterocycles 2002;57:1901-6.
  5. Karig G, Thasana N, Gallagher T. Directed deprotonation-transmetallation of 4-bromopyridine: flexible routes to substituted pyridines. Synlett 2002:808-10.
  6. Mahidol C, Kaweetripob W, Prawat H, Ruchirawat S. Mammea coumarins from the flowers of Mammea siamensis. J Nat Prod 2002;65:757-60.
  7. Mahidol C, Prawat H, Prachyawarakorn V, Ruchirawat S. Investigation of some bioactive thai medicinal plants. Phytochemistry Reviews 2002;1:287-97.
  8. Mahidol C, Prawat H, Kaweetripob W, Ruchirawat S. Two new pyranoflavanones from the stems of Derris reticulata. Heterocycles 2002;57:1287-92.
  9. Namsa-aid A, Ruchirawat S. Efficient synthesis of ningalin C. Org Lett 2002;4:2633-5.
  10. Siripong P, Nakamura ES, Kanokmedhakul K, Ruchirawat S, Saiki I. Anti-invasive effects of curcuminoid compounds from Curcuma aromatica Salisb. on murine colon 26-L5 carcinoma cells. J Trad Med 2002;19:209-15.
  11. Thasana N, Ruchirawat S. The application of the Baker–Venkataraman rearrangement to the synthesis of benz[b]indeno[2,1-e]pyran-10,11-dione. Tetrahedron Lett 2002;43:4515-7.
  12. Lirdprapamongkol K, Mahidol C, Thongnest S, Prawat H, Ruchirawat S, Srisomsap C, Surarit R, Punyarit P, Svasti J. Anti-metastatic effects of aqueous extract of Helixanthera parasitica. J Ethnopharmacol 2003;86:253-6.
  13. Ploypradith P, Jinaglueng W, Pavaro C, Ruchirawat S. Further developments in the synthesis of lamellarin alkaloids via direct metal–halogen exchange. Tetrahedron Lett 2003;44:1363-6.
  14. Ruchirawat S, Bhavakul V, Chaisupakitsin M. A one-pot synthesis of (±) cryptostylines I, II, III. Synth Commun 2003;33:621-5.
  15. Sahakitpichan P, Ruchirawat S. Highly efficient synthesis of buflavine: a unique Amaryllidaceae alkaloid. Tetrahedron Lett 2003;44:5239-41.
  16. Sutthivaiyakit S, Mongkolvisut W, Ponsitipiboon P, Prabpai S, Kongsaeree P, Ruchirawat S, Mahidol C. A novel 8,9-seco-rhamnofolane and a new rhamnofolane endoperoxide from Jatropha integerrima roots. Tetrahedron Lett 2003;44:3637-40.
  17. Thasana N, Ruchirawat S. The synthesis of wrightiadione via directed remote metalation. Synlett 2003:1037-9.
  18. Thasana N, Prachyawarakorn V, Tontoolarug S, Ruchirawat S. Synthesis of aryl α-keto esters via the rearrangement of aryl cyanohydrin carbonate esters. Tetrahedron Lett 2003;44:1019-21.
  19. Kanchanapoom T, Noiarsa P, Ruchirawat S, Kasai R, Otsuka H. Triterpenoidal glycosides from Justicia betonica. Phytochemistry 2004;65:2613-8.
  20. Kanchanapoom T, Ruchirawat S, Kasai R, Otsuka H. Aliphatic alcohol and iridoid glycosides from Asystasia intrusa. Chem Pharm Bull (Tokyo) 2004;52:980-2.
  21. Kanchanapoom T, Noiarsa P, Ruchirawat S, Kasai R, Otsuka H. Phenylethanoid and iridoid glycosides from the Thai medicinal plant, Barleria strigosa. Chem Pharm Bull (Tokyo) 2004;52:612-4.
  22. Pholphana N, Rangkadilok N, Thongnest S, Ruchirawat S, Ruchirawat M, Satayavivad J. Determination and variation of three active diterpenoids in Andrographis paniculata (Burm.f.) Nees. Phytochem Anal 2004;15:365-71.
  23. Ploypradith P, Mahidol C, Sahakitpichan P, Wongbundit S, Ruchirawat S. A highly efficient synthesis of lamellarins K and L by the Michael addition/ring-closure reaction of benzyldihydroisoquinoline derivatives with ethoxycarbonyl-β-nitrostyrenes. Angew Chem Int Ed Engl 2004;43:866-8.
  24. Sahakitpichan P, Ruchirawat S. A practical and highly efficient synthesis of lennoxamine and related isoindolobenzazepines. Tetrahedron 2004;60:4169-72.
  25. Satayavivad J, Watcharasit P, Khamkong P, Tuntawiroon J, Pavaro C, Ruchirawat S. The pharmacodynamic study of a potent new antimalarial (MC1). Acta Trop 2004;89:343-9.
  26. Kanchanapoom T, Noiarsa P, Tiengtham P, Otsuka H, Ruchirawat S. Acetophenone diglycosides from Erythroxylum cambodianum. Chem Pharm Bull (Tokyo) 2005;53:579-81.
  27. Kanchanapoom T, Noiarsa P, Ryoji K, Hideaki O, Ruchirawat S. Justiciosides E-G, triterpenoidal glycosides with an unusual skeleton from Justicia betonica. Tetrahedron 2005;61:2583-7.
  28. Lirdprapamongkol K, Sakurai H, Kawasaki N, Choo M-K, Saitoh Y, Aozuka Y, Singhirunnusorn P, Ruchirawat S, Svasti J, Saiki I. Vanillin suppresses in vitro invasion and in vivo metastasis of mouse breast cancer cells. Eur J Pharm Sci 2005;25:57-65.
  29. Phommart S, Sutthivaiyakit P, Chimnoi N, Ruchirawat S, Sutthivaiyakit S. Constituents of the leaves of Macaranga tanarius. J Nat Prod 2005;68:927-30.
  30. Ploypradith P, Kagan RK, Ruchirawat S. Utility of polymer-supported reagents in the total synthesis of lamellarins. J Org Chem 2005;70:5119-25.
  31. Sahakitpichan P, Thasana N, Ruchirawat S. Efficient synthesis of diospyrol via Suzuki–Miyaura and modified in situ cross-coupling. Synthesis 2005:2934-8.
  32. Suksamrarn S, Suwannapoch N, Aunchai N, Kuno M, Ratananukul P, Haritakun R, Jansakul C, Ruchirawat S. Ziziphine N, O, P and Q, new antiplasmodial cyclopeptide alkaloids from Ziziphus oenoplia var. brunoniana. Tetrahedron 2005;61:1175-80.
  33. Svasti J, Srisomsap C, Subhasitanont P, Keeratichamroen S, Chokchaichamnankit D, Ngiwsara L, Chimnoi N, Pisutjaroenpong S, Techasakul S, Chen S-T. Proteomic profiling of cholangiocarcinoma cell line treated with pomiferin from Derris malaccensis. Proteomics 2005;5:4504-9.
  34. Tempeam A, Thasana N, Pavaro C, Chuakul W, Siripong P, Ruchirawat S. A new cytotoxic daphnane diterpenoid, rediocide G, from Trigonostemon reidioides. Chem Pharm Bull (Tokyo) 2005;53:1321-3.
  35. Thongnest S, Mahidol C, Sutthivaiyakit S, Ruchirawat S. Oxygenated pimarane diterpenes from Kaempferia marginata. J Nat Prod 2005;68:1632-6.
  36. Athikomkulchai S, Prawat H, Thasana N, Ruangrungsi N, Ruchirawat S. COX-1, COX-2 inhibitors and antifungal agents from Croton hutchinsonianus. Chem Pharm Bull (Tokyo) 2006;54:262-4.
  37. Chomcheon P, Sriubolmas N, Wiyakrutta S, Ngamrojanavanich N, Chaichit N, Mahidol C, Ruchirawat S, Kittakoop P. Cyclopentenones, scaffolds for organic syntheses produced by the endophytic fungus mitosporic Dothideomycete sp. LRUB20. J Nat Prod 2006;69:1351-3.
  38. Kanchanapoom T, Sirikatitham A, Otsuka H, Ruchirawat S. Cuneatoside, a new megastigmane diglycoside from Erythroxylum cuneatum Blume. J Asian Nat Prod Res 2006;8:747-51.
  39. Kanchanapoom T, Noiarsa P, Otsuka H, Ruchirawat S. Lignan, phenolic and iridoid glycosides from Stereospermum cylindricum. Phytochemistry 2006;67:516-20.
  40. Kanchanapoom T, Noiarsa P, Otsuka H, Ruchirawat S. Chemical constituents of Acanthus volubilis Wall. Biochem Syst Ecol 2006;34:442-5.
  41. Likhitwitayawuid K, Sornsute A, Sritularak B, Ploypradith P. Chemical transformations of oxyresveratrol (trans-2,4,3',5'-tetrahydroxystilbene) into a potent tyrosinase inhibitor and a strong cytotoxic agent. Bioorg Med Chem Lett 2006;16:5650-3.
  42. Markmee S, Ruchirawat S, Prachyawarakorn V, Ingkaninan K, Khorana N. Isoquinoline derivatives as potential acetylcholinesterase inhibitors. Bioorg Med Chem Lett 2006;16:2170-2.
  43. Petchmanee T, Ploypradith P, Ruchirawat S. Solid-supported acids for debenzylation of aryl benzyl ethers. J Org Chem 2006;71:2892-5.
  44. Ploypradith P, Petchmanee T, Sahakitpichan P, Litvinas ND, Ruchirawat S. Total synthesis of natural and unnatural lamellarins with saturated and unsaturated D-rings. J Org Chem 2006;71:9440-8.
  45. Prachyawarakorn V, Mahidol C, Ruchirawat S. Siamenols A–D, four new coumarins from Mammea siamensis. Chem Pharm Bull (Tokyo) 2006;54:884-6.
  46. Prachyawarakorn V, Mahidol C, Ruchirawat S. Pyranocoumarins from the twigs of Mammea siamensis. Phytochemistry 2006;67:924-8.
  47. Siripong P, Yahuafai J, Shimizu K, Ichikawa K, Yonezawa S, Asai T, Kanokmedakul K, Ruchirawat S, Oku N. Antitumor activity of liposomal naphthoquinone esters isolated from Thai medicinal plant: Rhinacanthus nasutus KURZ. Biol Pharm Bull 2006;29:2279-83.
  48. Siripong P, Yahuafai J, Shimizu K, Ichikawa K, Yonezawa S, Asai T, Kanokmedakul K, Ruchirawat S, Oku N. Induction of apoptosis in tumor cells by three naphthoquinone esters isolated from Thai medicinal plant: Rhinacanthus nasutus KURZ. Biol Pharm Bull 2006;29:2070-6.
  49. Thasana N, Pisutjaroenpong S, Ruchirawat S. Two protocols for the conversion of biphenol to binaphthol: synthesis of diospyrol. Synlett 2006:1080-4.
  50. Thisoda P, Rangkadilok N, Pholphana N, Worasuttayangkurn L, Ruchirawat S, Satayavivad J. Inhibitory effect of Andrographis paniculata extract and its active diterpenoids on platelet aggregation. Eur J Pharmacol 2006;553:39-45.
  51. Worayuthakarn R, Thasana N, Ruchirawat S. Three distinct reactions of 3,4-dihydroisoquinolines with azlactones: novel synthesis of imidazoloisoquinolin-3-ones, benzo[α]quinolizin-4-ones, and benzo[d]azocin-4-ones. Org Lett 2006;8:5845-8.
  52. Boonphong S, Puangsombat P, Baramee A, Mahidol C, Ruchirawat S, Kittakoop P. Bioactive compounds from Bauhinia purpurea possessing antimalarial, antimycobacterial, antifungal, anti-inflammatory, and cytotoxic activities. J Nat Prod 2007;70:795-801.
  53. Ploypradith P, Cheryklin P, Niyomtham N, Bertoni DR, Ruchirawat S. Solid-supported acids as mild and versatile reagents for the deprotection of aromatic ethers. Org Lett 2007;9:2637-40.
  54. Yoopan N, Thisoda P, Rangkadilok N, Sahasitiwat S, Pholphana N, Ruchirawat S, Satayavivad J. Cardiovascular effects of 14-deoxy-11,12-didehydroandrographolide and Andrographis paniculata extracts. Planta Med 2007;73:503-11.
  55. Kanchanapoom T, Otsuka H, Ruchirawat S. Megastigmane glucosides from Equisetum debile and E. diffusum. Chem Pharm Bull (Tokyo) 2007;55:1277-80.
  56. Prachya S, Wiyakrutta S, Sriubolmas N, Ngamrojanavanich N, Mahidol C, Ruchirawat S, Kittakoop P. Cytotoxic mycoepoxydiene derivatives from an endophytic fungus Phomopsis sp. isolated from Hydnocarpus anthelminthicus. Planta Med 2007;73:1418-20.
  57. Youngsa-ad W, Ngamrojanavanich N, Mahidol C, Ruchirawat S, Prawat H, Kittakoop P. Diterpenoids from the roots of Croton oblongifolius. Planta Med 2007;73:1491-4.
  58. Thasana N, Worayuthakarn R, Kradanrat P, Hohn E, Young L, Ruchirawat S. Copper(I)-Mediated and Microwave-Assisted Caryl-Ocarboxylic Coupling: Synthesis of Benzopyaranones and Isolamellarin Alkaloids. J Org Chem 2007;72:9379-82.
  59. Prachyawarakorn V, Mahidol C, Sureram S, Sangpetsiripan S, Wiyakrutta S, Ruchirawat S, Kittakoop P. Diketopiperazines and phthalides from a marine derived fungus of the order Pleosporales. Planta Med 2008; in press.
  60. Thasana N, Bjerke-Kroll B, Ruchirawat S. A facile synthesis of telisatin A via microwave-promoted annulation and Reformatsky reaction. Synlett 2008, accepted.

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